five

PDE2 catalytic domain complexed with inhibitors

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Protein Data Bank Japan2023-10-04 更新2026-03-21 收录
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PDE2 catalytic domain complexed with inhibitors Descriptor: 4-[3-(4-methoxyphenoxy)azetidin-1-yl]-1-methyl-3-(2-methylpropyl)-1H-pyrazolo[3,4-d]pyrimidine, MAGNESIUM ION, ZINC ION, ... Authors: Pandit, J. Deposit date: 2016-12-12 Release date: 2017-06-28 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (2 Å) Cite: Application of Structure-Based Design and Parallel Chemistry to Identify a Potent, Selective, and Brain Penetrant Phosphodiesterase 2A Inhibitor. J. Med. Chem., 60, 2017
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2016-12-12
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