five

Discovery of phenoxyindazoles and phenylthioindazoles as RORg inverse agonists

收藏
Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/5lwp
下载链接
链接失效反馈
官方服务:
资源简介:
Discovery of phenoxyindazoles and phenylthioindazoles as RORg inverse agonists Descriptor: 4-[3-[2-chloranyl-6-(trifluoromethyl)phenoxy]-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid, Nuclear receptor ROR-gamma Authors: Ouvry, G, Bouix-Peter, C, Ciesielski, F, Chantalat, L, Christin, O, Comino, C, Duvert, D, Feret, C, Harris, C.S, Luzy, A.-P, Musicki, B, Orfila, D, Pascau, J, Parnet, V, Perrin, A, Pierre, R, Raffin, C, Rival, Y, Taquet, N, Thoreau, E, Hennequin, L.F. Deposit date: 2016-09-19 Release date: 2016-11-16 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Discovery of phenoxyindazoles and phenylthioindazoles as ROR gamma inverse agonists. Bioorg.Med.Chem.Lett., 26, 2016
创建时间:
2016-09-19
二维码
社区交流群
二维码
科研交流群
商业服务