CRYSTAL STRUCTURE OF NATIVE HUMAN MYELOPEROXIDASE IN COMPLEX WITH CPD 3
收藏Protein Data Bank Japan2024-11-20 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7ni3
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CRYSTAL STRUCTURE OF NATIVE HUMAN MYELOPEROXIDASE IN COMPLEX WITH CPD 3 Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-sulfanylidene-3-[(2R)-tetrahydro-2-furanylmethyl]-1,2,3,7-tetrahydro-6H-purin-6-one, CALCIUM ION, ... Authors: Sjogren, T, Inghardt, T. Deposit date: 2021-02-11 Release date: 2022-02-23 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Discovery of AZD4831, a Mechanism-Based Irreversible Inhibitor of Myeloperoxidase, As a Potential Treatment for Heart Failure with Preserved Ejection Fraction. J.Med.Chem., 65, 2022
创建时间:
2021-02-11



