Crystal Structure of the first bromodomain of human BRD4 in complex with the inhibitor TG-101348
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Crystal Structure of the first bromodomain of human BRD4 in complex with the inhibitor TG-101348 Descriptor: 1,2-ETHANEDIOL, Bromodomain-containing protein 4, N-tert-butyl-3-{[5-methyl-2-({4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}amino)pyrimidin-4-yl]amino}benzenesulfonamide Authors: Filippakopoulos, P, Picaud, S, Jose, B, Martin, S, Fedorov, O, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2014-01-16 Release date: 2014-02-26 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (1.65 Å) Cite: Dual kinase-bromodomain inhibitors for rationally designed polypharmacology. Nat.Chem.Biol., 10, 2014
创建时间：
2014-01-16
