Tankyrase 2 in complex with an inhibitor (OM-1800)
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Tankyrase 2 in complex with an inhibitor (OM-1800) Descriptor: Tankyrase-2, ZINC ION, ~{N}-[3-[5-(5-ethoxypyridin-2-yl)-4-(2-fluorophenyl)-1,2,4-triazol-3-yl]cyclobutyl]-1,5-naphthyridine-4-carboxamide Authors: Sowa, S.T, Lehtio, L. Deposit date: 2019-11-28 Release date: 2020-07-08 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.7 Å) Cite: Preclinical Lead Optimization of a 1,2,4-Triazole Based Tankyrase Inhibitor. J.Med.Chem., 63, 2020
创建时间:
2019-11-28



