Crystal structure of human pyruvate dehydrogenase kinase 4 in complex with compound 7
收藏Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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Crystal structure of human pyruvate dehydrogenase kinase 4 in complex with compound 7 Descriptor: 3,3-dimethyl-7-(methylamino)-1H-indol-2-one, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... Authors: Orita, T, Doi, S, Iwanaga, T, Adachi, T. Deposit date: 2021-03-09 Release date: 2021-08-04 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Fragment-based lead discovery to identify novel inhibitors that target the ATP binding site of pyruvate dehydrogenase kinases. Bioorg.Med.Chem., 44, 2021
创建时间:
2021-03-09



