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Src kinase bound to eCF506 trapped in inactive conformation

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Protein Data Bank Japan2024-01-31 更新2026-04-19 收录
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资源简介:
Src kinase bound to eCF506 trapped in inactive conformation Descriptor: 1,2-ETHANEDIOL, Proto-oncogene tyrosine-protein kinase Src, tert-butyl (4-(4-amino-1-(2-(4-(dimethylamino)piperidin-1-yl)ethyl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)carbamate Authors: Lietha, D, Unciti-Broceta, A. Deposit date: 2021-02-08 Release date: 2021-09-15 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.5 Å) Cite: A Conformation Selective Mode of Inhibiting SRC Improves Drug Efficacy and Tolerability. Cancer Res., 81, 2021
创建时间:
2021-02-08
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