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Crystal structure of G238A mutant of TEM-1 beta-lactamase in complex with a boronic acid inhibitor (sefb4)

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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Crystal structure of G238A mutant of TEM-1 beta-lactamase in complex with a boronic acid inhibitor (sefb4) Descriptor: BETA-LACTAMASE TEM, PINACOL[[2-AMINO-ALPHA-(1-CARBOXY-1-METHYLETHOXYIMINO)-4-THIAZOLEACETYL]AMINO]METHANEBORONATE, POTASSIUM ION Authors: Wang, X, Minasov, G, Shoichet, B.K. Deposit date: 2001-09-05 Release date: 2002-06-05 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Evolution of an antibiotic resistance enzyme constrained by stability and activity trade-offs. J.Mol.Biol., 320, 2002
创建时间:
2001-09-05
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