five

C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 5-(1-benzyl-4-chloro-1H-imidazol-2-yl)-1,3-dimethylpyridin-2(1H)-one

收藏
Protein Data Bank Japan2024-07-10 更新2026-05-23 收录
下载链接:
https://pdbj.org/mine/summary/9fbx
下载链接
链接失效反馈
官方服务:
资源简介:
C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 5-(1-benzyl-4-chloro-1H-imidazol-2-yl)-1,3-dimethylpyridin-2(1H)-one Descriptor: 1,2-ETHANEDIOL, 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, 5-(1-benzyl-4-chloro-1H-imidazol-2-yl)-1,3-dimethylpyridin-2(1H)-one, ... Authors: Chung, C. Deposit date: 2024-05-14 Release date: 2024-06-26 Last modified: 2024-07-10 Method: X-RAY DIFFRACTION (1.602 Å) Cite: Structure- and Property-Based Optimization of Efficient Pan-Bromodomain and Extra Terminal Inhibitors to Identify Oral and Intravenous Candidate I-BET787. J.Med.Chem., 67, 2024
创建时间:
2024-05-14
二维码
社区交流群
二维码
科研交流群
商业服务