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Crystal structure of PI3K-gamma in complex with triazine-benzimidazole 32

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Protein Data Bank Japan2023-09-13 更新2026-03-21 收录
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Crystal structure of PI3K-gamma in complex with triazine-benzimidazole 32 Descriptor: 1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(1H-pyrazol-3-yl)-1H-benzimidazol-2-amine, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, SULFATE ION Authors: Whittington, D.A, Tang, J, Yakowec, P. Deposit date: 2011-01-11 Release date: 2011-03-30 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (2.65 Å) Cite: Discovery of triazine-benzimidazoles as selective inhibitors of mTOR. Bioorg.Med.Chem.Lett., 21, 2011

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2011-01-11
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