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ACE2 in complex with bicyclic peptide inhibitor

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Protein Data Bank Japan2026-03-04 更新2026-04-25 收录
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ACE2 in complex with bicyclic peptide inhibitor Descriptor: 1-[3,5-bis(3-bromanylpropanoyl)-1,3,5-triazinan-1-yl]-3-bromanyl-propan-1-one, ALA-CYS-GLY-ARG-GLN-PHE-CYS-HIS-THR-LEU-MET-PRO-ARG-HIS-LEU-CYS-ALA-NH2, Processed angiotensin-converting enzyme 2 Authors: Brear, P, Lulla, A, Harman, M, Dods, R, Chen, L, Bezerra, G, Demydchuk, Y, Stanway, S, Hyvonen, M. Deposit date: 2022-10-06 Release date: 2023-09-20 Last modified: 2026-03-04 Method: X-RAY DIFFRACTION (2.11 Å) Cite: Structure-Guided Chemical Optimization of Bicyclic Peptide ( Bicycle ) Inhibitors of Angiotensin-Converting Enzyme 2. J.Med.Chem., 66, 2023
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2022-10-06
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