Crystal structure of the human BRPF1 bromodomain in complex with BZ135
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Crystal structure of the human BRPF1 bromodomain in complex with BZ135 Descriptor: NITRATE ION, Peregrin, ~{N}-[1,4-dimethyl-7-morpholin-4-yl-2,3-bis(oxidanylidene)quinoxalin-6-yl]-5,6,7,8-tetrahydronaphthalene-2-sulfonamide Authors: Zhu, J, Caflisch, A. Deposit date: 2017-05-30 Release date: 2018-06-13 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.75 Å) Cite: Structure-based discovery of selective BRPF1 bromodomain inhibitors. Eur J Med Chem, 155, 2018
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2017-05-30



