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Discovery of an Orally Biovailable KRAS G12D Inhibitor

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Protein Data Bank Japan2025-02-05 更新2026-08-24 收录
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Discovery of an Orally Biovailable KRAS G12D Inhibitor Descriptor: GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... Authors: Deller, M.C, Epling, L.B. Deposit date: 2024-10-28 Release date: 2025-01-22 Last modified: 2025-02-05 Method: X-RAY DIFFRACTION (1.36 Å) Cite: Discovery of INCB159020, an Orally Bioavailable KRAS G12D Inhibitor. J.Med.Chem., 68, 2025

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2024-10-28
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