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Human MTHFD2 in complex with DS44960156

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Protein Data Bank Japan2023-11-22 更新2026-03-21 收录
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Human MTHFD2 in complex with DS44960156 Descriptor: 4-(5-oxo-1,5-dihydro-2H-[1]benzopyrano[3,4-c]pyridine-3(4H)-carbonyl)benzoic acid, Bifunctional methylenetetrahydrofolate dehydrogenase/cyclohydrolase, mitochondrial, ... Authors: Suzuki, M, Matsui, Y, Kawai, J. Deposit date: 2019-02-20 Release date: 2019-06-05 Last modified: 2023-11-22 Method: X-RAY DIFFRACTION (2.25 Å) Cite: Structure-Based Design and Synthesis of an Isozyme-Selective MTHFD2 Inhibitor with a Tricyclic Coumarin Scaffold. Acs Med.Chem.Lett., 10, 2019
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2019-02-20
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