Crystal structure of pyruvate dehydrogenase kinase isoform 2 in complex with inhibitor PA1
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Crystal structure of pyruvate dehydrogenase kinase isoform 2 in complex with inhibitor PA1 Descriptor: (5-bromo-2,4-dihydroxyphenyl)(1,3-dihydro-2H-isoindol-2-yl)methanone, L(+)-TARTARIC ACID, [Pyruvate dehydrogenase [lipoamide]] kinase isozyme 2, ... Authors: Gui, W.J, Tso, S.C, Chuang, J.L, Wu, C.Y, Qi, X, Tambar, U.K, Wynn, R.M, Chuang, D.T. Deposit date: 2013-09-12 Release date: 2014-01-01 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (1.751 Å) Cite: Structure-guided Development of Specific Pyruvate Dehydrogenase Kinase Inhibitors Targeting the ATP-binding Pocket. J.Biol.Chem., 289, 2014
创建时间:
2013-09-12



