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CRYSTAL STRUCTURE OF PHD2 CATALYTIC DOMAIN (CID 7465) IN COMPLEX WITH AKB-6548 AT 1.8 A RESOLUTION

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Protein Data Bank Japan2023-10-25 更新2026-03-28 收录
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CRYSTAL STRUCTURE OF PHD2 CATALYTIC DOMAIN (CID 7465) IN COMPLEX WITH AKB-6548 AT 1.8 A RESOLUTION Descriptor: 1,2-ETHANEDIOL, Egl nine homolog 1, FE (II) ION, ... Authors: Davie, D.R, Abendroth, J, Boyd, J. Deposit date: 2022-04-07 Release date: 2022-05-18 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Preclinical Characterization of Vadadustat (AKB-6548), an Oral Small Molecule Hypoxia-Inducible Factor Prolyl-4-Hydroxylase Inhibitor, for the Potential Treatment of Renal Anemia. J.Pharmacol.Exp.Ther., 383, 2022
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2022-04-07
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