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HUMAN PI3KDELTA IN COMPLEX WITH COMPOUND 2F

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Protein Data Bank Japan2024-04-03 更新2026-03-28 收录
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https://pdbj.org/mine/summary/7jiu
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HUMAN PI3KDELTA IN COMPLEX WITH COMPOUND 2F Descriptor: (3S)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9H-purin-6-yl]-3-methyl-1,3-dihydro-2H-indol-2-one, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform Authors: Lesburg, C.A, Augustin, M. Deposit date: 2020-07-23 Release date: 2021-06-30 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2.12 Å) Cite: Optimization of Versatile Oxindoles as Selective PI3K delta Inhibitors. Acs Med.Chem.Lett., 11, 2020
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2020-07-23
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