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Crystal structure of the first bromodomain (BD1) of human BRD3 bound to SG3-179

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Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Crystal structure of the first bromodomain (BD1) of human BRD3 bound to SG3-179 Descriptor: 1,2-ETHANEDIOL, 4-[[4-[[3-(~{tert}-butylsulfonylamino)-4-chloranyl-phenyl]amino]-5-methyl-pyrimidin-2-yl]amino]-2-fluoranyl-~{N}-(1-methylpiperidin-4-yl)benzamide, Bromodomain-containing protein 3, ... Authors: Karim, M.R, Bikowitz, M.J, Schonbrunn, E. Deposit date: 2021-01-07 Release date: 2021-07-14 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.45 Å) Cite: Differential BET Bromodomain Inhibition by Dihydropteridinone and Pyrimidodiazepinone Kinase Inhibitors. J.Med.Chem., 64, 2021
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2021-01-07
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