AmpC beta-lactamase in complex with 3-(4-carboxy-2-hydroxy-phenylsulfamoyl)-thiophene-2-carboxylic acid
收藏Protein Data Bank Japan2023-08-23 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/1xgj
下载链接
链接失效反馈官方服务:
资源简介:
AmpC beta-lactamase in complex with 3-(4-carboxy-2-hydroxy-phenylsulfamoyl)-thiophene-2-carboxylic acid Descriptor: 3-{[(4-CARBOXY-2-HYDROXYANILINE]SULFONYL}THIOPHENE-2-CARBOXYLIC ACID, Beta-lactamase Authors: Tondi, D, Morandi, F, Bonnet, R, Costi, M.P, Shoichet, B.K. Deposit date: 2004-09-17 Release date: 2005-05-03 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (1.97 Å) Cite: Structure-based optimization of a non-beta-lactam lead results in inhibitors that do not up-regulate beta-lactamase expression in cell culture. J.Am.Chem.Soc., 127, 2005
创建时间:
2004-09-17



