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IRAK4 in complex with inhibitor

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Protein Data Bank Japan2024-10-16 更新2026-04-19 收录
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IRAK4 in complex with inhibitor Descriptor: 6-methyl-4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[4,3-d]pyrimidin-5-one, Interleukin-1 receptor-associated kinase 4 Authors: Xue, Y, Aagaard, A, Robb, G.R, Degorce, S.L. Deposit date: 2021-12-07 Release date: 2022-05-04 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (3.031 Å) Cite: Identification and optimisation of a pyrimidopyridone series of IRAK4 inhibitors. Bioorg.Med.Chem., 63, 2022

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2021-12-07
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