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Calpain 1 proteolytic core in complex with SNJ-1945, a alpha-ketoamide-type inhibitor.

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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Calpain 1 proteolytic core in complex with SNJ-1945, a alpha-ketoamide-type inhibitor. Descriptor: ((1S)-1-((((1S)-1-BENZYL-3-(CYCLOPROPYLAMINO)-2,3-DIOXOPROPYL)AMINO)CARBONYL)-3-METHYLBUTYL)CARBAMIC ACID 5-METHOXY-3-OXAPENTYL ESTER, CALCIUM ION, Calpain-1 catalytic subunit Authors: Cuerrier, D, Moldoveanu, T, Davies, P.L, Campbell, R.L. Deposit date: 2006-03-02 Release date: 2006-06-06 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (1.61 Å) Cite: Calpain Inhibition by alpha-Ketoamide and Cyclic Hemiacetal Inhibitors Revealed by X-ray Crystallography Biochemistry, 45, 2006

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2006-03-02
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