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The Influence of I47A Mutation on Reduced Susceptibility to the Protease Inhibitor Lopinavir

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Protein Data Bank Japan2023-08-30 更新2026-03-21 收录
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The Influence of I47A Mutation on Reduced Susceptibility to the Protease Inhibitor Lopinavir Descriptor: BETA-MERCAPTOETHANOL, N-{1-BENZYL-4-[2-(2,6-DIMETHYL-PHENOXY)-ACETYLAMINO]-3-HYDROXY-5-PHENYL-PENTYL}-3-METHYL-2-(2-OXO-TETRAHYDRO-PYRIMIDIN-1-YL)-BUTYRAMIDE, PROTEASE RETROPEPSIN Authors: Brynda, J, Saskova, K.G, Kozisek, M, Lepsik, M, Machala, L, Konvalinka, J. Deposit date: 2007-07-02 Release date: 2008-07-22 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (2.802 Å) Cite: Enzymatic and structural analysis of the I47A mutation contributing to the reduced susceptibility to HIV protease inhibitor lopinavir. Protein Sci., 17, 2008
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2007-07-02
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