Catalytic domain of human phosphodiesterase 4B2B in complex with a quinoline inhibitor
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Catalytic domain of human phosphodiesterase 4B2B in complex with a quinoline inhibitor Descriptor: 6-{[3-(dimethylcarbamoyl)phenyl]sulfonyl}-4-[(3-methoxyphenyl)amino]-8-methylquinoline-3-carboxamide, ARSENIC, GLYCEROL, ... Authors: Somers, D.O, Neu, M. Deposit date: 2009-04-01 Release date: 2010-04-07 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (1.75 Å) Cite: Quinolines as a novel structural class of potent and selective PDE4 inhibitors. Optimisation for inhaled administration. Bioorg.Med.Chem.Lett., 19, 2009
创建时间:
2009-04-01



