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Crystal structure of CK1 delta in complex with VN725

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Protein Data Bank Japan2024-02-07 更新2026-04-25 收录
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Crystal structure of CK1 delta in complex with VN725 Descriptor: 1,2-ETHANEDIOL, 4-[3-cyclohexyl-5-(4-fluorophenyl)imidazol-4-yl]-1~{H}-pyrrolo[2,3-b]pyridine, Casein kinase I isoform delta, ... Authors: Chaikuad, A, Nemec, V, Paruch, K, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2022-01-10 Release date: 2023-01-18 Last modified: 2024-02-07 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Discovery of Potent and Exquisitely Selective Inhibitors of Kinase CK1 with Tunable Isoform Selectivity. Angew.Chem.Int.Ed.Engl., 62, 2023

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2022-01-10
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