遇见数据集

KRAS-169 Q61H GPPNHP + PPIN-1

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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KRAS-169 Q61H GPPNHP + PPIN-1 Descriptor: (6~{S})-1-(1~{H}-imidazol-4-ylcarbonyl)-6-[(4-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one, CITRIC ACID, GTPase KRas, ... Authors: Cruz-Migoni, A, Canning, P, Quevedo, C.E, Carr, S.B, Phillips, S.E.V, Rabbitts, T.H. Deposit date: 2018-06-01 Release date: 2019-02-06 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (1.63 Å) Cite: Structure-based development of new RAS-effector inhibitors from a combination of active and inactive RAS-binding compounds. Proc. Natl. Acad. Sci. U.S.A., 116, 2019

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2018-06-01
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