five

CARM1 bound with compound 43

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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CARM1 bound with compound 43 Descriptor: Histone-arginine methyltransferase CARM1, N'-[[3-[4-(3,5-dimethyl-1,2-oxazol-4-yl)-5-methyl-6-phenylazanyl-pyrimidin-2-yl]phenyl]methyl]-N-methyl-ethane-1,2-diamine Authors: Cao, D.Y, Li, J, Xiong, B. Deposit date: 2021-07-06 Release date: 2021-11-24 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (2.24507255823 Å) Cite: Structure-Based Discovery of Potent CARM1 Inhibitors for Solid Tumor and Cancer Immunology Therapy. J.Med.Chem., 64, 2021
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2021-07-06
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