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Crystal structure of Candida glabrata Bdf1 bromodomain 1 bound to a pyrazole ligand

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Protein Data Bank Japan2025-03-26 更新2026-04-19 收录
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Crystal structure of Candida glabrata Bdf1 bromodomain 1 bound to a pyrazole ligand Descriptor: 2-methyl-~{N}-[[5-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)thiophen-2-yl]methyl]pyrazole-3-carboxamide, Candida glabrata strain CBS138 chromosome C complete sequence, SULFATE ION Authors: Petosa, C, Wei, K, McKenna, C.E, Govin, J. Deposit date: 2023-11-22 Release date: 2024-10-30 Last modified: 2025-03-26 Method: X-RAY DIFFRACTION (1.82 Å) Cite: Humanized Candida and NanoBiT Assays Expedite Discovery of Bdf1 Bromodomain Inhibitors With Antifungal Potential. Adv Sci, 12, 2025
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2023-11-22
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