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Human PARP14 (ARTD8), catalytic fragment in complex with RBN012042

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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Human PARP14 (ARTD8), catalytic fragment in complex with RBN012042 Descriptor: 1,2-ETHANEDIOL, 7-(cyclopentylamino)-5-fluoro-2-{[(piperidin-4-yl)sulfanyl]methyl}quinazolin-4(3H)-one, CHLORIDE ION, ... Authors: Dorsey, B.W, Swinger, K.K, Schenkel, L.B, Church, W.D, Perl, N.R, Vasbinder, M.M, Wigle, T.J, Kuntz, K.W. Deposit date: 2021-01-05 Release date: 2021-04-21 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.25 Å) Cite: Targeted Degradation of PARP14 Using a Heterobifunctional Small Molecule. Chembiochem, 22, 2021

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2021-01-05
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