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Cannabinoid receptor 1-Gi complex with novel ligand

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Protein Data Bank Japan2025-05-07 更新2026-04-19 收录
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https://pdbj.org/mine/summary/9dgi
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Cannabinoid receptor 1-Gi complex with novel ligand Descriptor: Cannabinoid receptor 1, methyl (2R)-2-({(1M)-5-methyl-1-[3-(trifluoromethyl)phenyl]-1H-pyrazole-3-carbonyl}amino)-2-(thiophen-2-yl)propanoate Authors: Tummino, T.A, Iliopoulos-Tsoutsouvas, C, Braz, J.M, O'Brien, E.S, Krishna Kumar, K, Makriyannis, M, Basbaum, A.I, Shoichet, B.K. Deposit date: 2024-09-02 Release date: 2025-04-30 Last modified: 2025-05-07 Method: ELECTRON MICROSCOPY (3.35 Å) Cite: Virtual library docking for cannabinoid-1 receptor agonists with reduced side effects. Nat Commun, 16, 2025
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2024-09-02
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