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Crystal structure of PDE10A in complex with a triazolopyrimidine inhibitor

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Protein Data Bank Japan2023-11-22 更新2026-03-21 收录
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Crystal structure of PDE10A in complex with a triazolopyrimidine inhibitor Descriptor: 2-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-1-[(2S)-2-methyl-1,2-dihydroimidazo[1,2-a]benzimidazol-3-yl]ethanone, MAGNESIUM ION, ZINC ION, ... Authors: Amano, Y, Honbou, K. Deposit date: 2019-07-03 Release date: 2019-08-14 Last modified: 2023-11-22 Method: X-RAY DIFFRACTION (2.95 Å) Cite: Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors. Bioorg.Med.Chem., 27, 2019

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2019-07-03
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