Tricyclic indazoles a novel class of selective estrogen receptor degrader antagonists
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Tricyclic indazoles a novel class of selective estrogen receptor degrader antagonists Descriptor: 3-[4-[(6~{R})-7-(2-methylpropyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]phenyl]propanoic acid, Estrogen receptor Authors: Scott, J.S, Bailey, A, Buttar, D, Carbajo, R.J, Curwen, J, Davies, R.D.M, Degorce, S.L, Donald, C, Gangl, E, Greenwood, R, Groombridge, S.D, Johnson, T, Lamont, S, Lawson, M, Lister, A, Morrow, C, Moss, T, Pink, J.H, Polanski, R. Deposit date: 2018-11-27 Release date: 2019-01-23 Last modified: 2024-05-15 Method: X-RAY DIFFRACTION (1.84 Å) Cite: Tricyclic Indazoles-A Novel Class of Selective Estrogen Receptor Degrader Antagonists. J.Med.Chem., 62, 2019
创建时间:
2018-11-27



