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Abl kinase in complex with imatinib and fragment (FRAG2) in the myristate site

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Protein Data Bank Japan2023-09-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/3mss
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Abl kinase in complex with imatinib and fragment (FRAG2) in the myristate site Descriptor: 4-(4-METHYL-PIPERAZIN-1-YLMETHYL)-N-[4-METHYL-3-(4-PYRIDIN-3-YL-PYRIMIDIN-2-YLAMINO)-PHENYL]-BENZAMIDE, O-benzyl-N-methyl-L-tyrosinamide, Tyrosine-protein kinase ABL1 Authors: Cowan-Jacob, S.W, Rummel, G, Fendrich, G. Deposit date: 2010-04-29 Release date: 2010-05-26 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Binding or bending: distinction of allosteric Abl kinase agonists from antagonists by an NMR-based conformational assay. J.Am.Chem.Soc., 132, 2010
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2010-04-29
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