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Covalent and non-covalent inhibitor of ERK2 (two sites)

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Protein Data Bank Japan2024-11-20 更新2026-03-28 收录
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https://pdbj.org/mine/summary/8aoa
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Covalent and non-covalent inhibitor of ERK2 (two sites) Descriptor: 1,2-ETHANEDIOL, DIMETHYL SULFOXIDE, Mitogen-activated protein kinase 1, ... Authors: Cleasby, A. Deposit date: 2022-08-08 Release date: 2022-09-28 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.62 Å) Cite: X-ray Screening of an Electrophilic Fragment Library and Application toward the Development of a Novel ERK 1/2 Covalent Inhibitor. J.Med.Chem., 65, 2022
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2022-08-08
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