遇见数据集

CK2 alpha bound to Macrocycle

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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CK2 alpha bound to Macrocycle Descriptor: 7,10-Dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid, Casein kinase II subunit alpha, SULFATE ION Authors: Kraemer, A, Hanke, T, Kurz, C, Celik, I, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2020-04-27 Release date: 2020-07-01 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Optimization of pyrazolo[1,5-a]pyrimidines lead to the identification of a highly selective casein kinase 2 inhibitor. Eur.J.Med.Chem., 208, 2020

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2020-04-27
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