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P38 alpha kinase complexed with a pyrazolo-pyrimidine based inhibitor

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Protein Data Bank Japan2024-02-21 更新2026-03-21 收录
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https://pdbj.org/mine/summary/3l8x
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P38 alpha kinase complexed with a pyrazolo-pyrimidine based inhibitor Descriptor: Mitogen-activated protein kinase 14, N,4-dimethyl-3-[(1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide Authors: Sack, J.S. Deposit date: 2010-01-04 Release date: 2010-03-02 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Pyrazolo-Pyrimidines: A Novel Heterocyclic Scaffold for Potent and Selective P38 Alpha Inhibitors. Bioorg.Med.Chem.Lett., 18, 2008
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2010-01-04
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