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Crystal structure of Rock1 with a pyridinylbenzamide based inhibitor

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Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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Crystal structure of Rock1 with a pyridinylbenzamide based inhibitor Descriptor: N-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamide, Rho-associated protein kinase 1, SULFATE ION Authors: Judge, R.A, Hobson, A.D. Deposit date: 2018-08-01 Release date: 2018-11-14 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.96 Å) Cite: Identification of Selective Dual ROCK1 and ROCK2 Inhibitors Using Structure Based Drug Design. J. Med. Chem., 61, 2018
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2018-08-01
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