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The Estrogen Receptor Alpha Ligand Binding Domain D538G Mutant in Complex with 4-hydroxytamoxifen

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Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4q50
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资源简介:
The Estrogen Receptor Alpha Ligand Binding Domain D538G Mutant in Complex with 4-hydroxytamoxifen Descriptor: 4-HYDROXYTAMOXIFEN, Estrogen receptor, SULFATE ION Authors: Fanning, S.W, Greene, G.L. Deposit date: 2014-04-15 Release date: 2015-04-15 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (3.07 Å) Cite: Estrogen receptor alpha somatic mutations Y537S and D538G confer breast cancer endocrine resistance by stabilizing the activating function-2 binding conformation. Elife, 5, 2016
创建时间:
2014-04-15
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