Crystal Structure of the first bromodomain of human BRD4 in complex with a isoxazolylbenzimidazole ligand
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Crystal Structure of the first bromodomain of human BRD4 in complex with a isoxazolylbenzimidazole ligand Descriptor: (1R)-6-(3,5-dimethyl-1,2-oxazol-4-yl)-1-phenyl-2,3-dihydro-1H-inden-1-ol, 1,2-ETHANEDIOL, Bromodomain-containing protein 4, ... Authors: Filippakopoulos, P, Picaud, S, Qi, J, Felletar, I, Heightman, T.D, Brennan, P, von Delft, F, Bountra, C, Arrowsmith, C.H, Edwards, A, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2012-08-21 Release date: 2012-10-17 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (1.6 Å) Cite: The design and synthesis of 5- and 6-isoxazolylbenzimidazoles as selective inhibitors of the BET bromodomains. Medchemcomm, 4, 2013
创建时间：
2012-08-21
