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Crystal Structure of Aurora-A in complex with a new Quinazoline inhibitor

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Protein Data Bank Japan2025-09-24 更新2026-03-21 收录
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Crystal Structure of Aurora-A in complex with a new Quinazoline inhibitor Descriptor: 7-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]quinazolin-4-amine, Aurora kinase A Authors: Cheng, B, Lu, G, Zhou, H. Deposit date: 2018-02-07 Release date: 2019-02-13 Last modified: 2025-09-24 Method: X-RAY DIFFRACTION (2.85 Å) Cite: Optimization of Novel Quinazolines as Potent Aurora Kinase Inhibitors for Triple-Negative Breast Cancer Treatment. J.Med.Chem., 68, 2025
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2018-02-07
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