AURORA KINASE A IN COMPLEX WITH THE AUR-A/PDK1 INHIBITOR VI8
收藏Protein Data Bank Japan2024-01-31 更新2026-03-28 收录
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AURORA KINASE A IN COMPLEX WITH THE AUR-A/PDK1 INHIBITOR VI8 Descriptor: 1-[[3,4-bis(fluoranyl)phenyl]methyl]-~{N}-[(1~{R})-2-[[(3~{E})-3-(1~{H}-imidazol-5-ylmethylidene)-2-oxidanylidene-1~{H}-indol-5-yl]amino]-2-oxidanylidene-1-phenyl-ethyl]-6-methyl-2-oxidanylidene-pyridine-3-carboxamide, Aurora kinase A Authors: Garau, G. Deposit date: 2021-03-31 Release date: 2021-10-20 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (3.1 Å) Cite: Development of potent dual PDK1/AurA kinase inhibitors for cancer therapy: Lead-optimization, structural insights, and ADME-Tox profile. Eur.J.Med.Chem., 226, 2021
创建时间：
2021-03-31
