Structure of cIAP1 with BCCov
收藏Protein Data Bank Japan2024-05-01 更新2026-04-25 收录
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Structure of cIAP1 with BCCov Descriptor: (4S)-4-[2-(2-{4-[(2E)-4-{(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}-4-oxobut-2-en-1-yl]piperazin-1-yl}ethoxy)acetamido]-1-{(2S)-2-cyclohexyl-2-[(N-methyl-L-alanyl)amino]acetyl}-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-L-prolinamide unbound form, Baculoviral IAP repeat-containing protein 2, ZINC ION Authors: Schiemer, J.S, Calabrese, M.F. Deposit date: 2022-07-22 Release date: 2023-03-08 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.5 Å) Cite: A covalent BTK ternary complex compatible with targeted protein degradation. Nat Commun, 14, 2023
创建时间:
2022-07-22



