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Crystal Structure of KPT8602 in complex with CRM1-Ran-RanBP1

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Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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Crystal Structure of KPT8602 in complex with CRM1-Ran-RanBP1 Descriptor: (2R)-3-{3-[3,5-bis(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}-2-(pyrimidin-5-yl)propanamide, CHLORIDE ION, Exportin-1, ... Authors: Fung, H.Y, Chook, Y.M. Deposit date: 2016-04-27 Release date: 2016-06-29 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (2.5 Å) Cite: Next-generation XPO1 inhibitor shows improved efficacy and in vivo tolerability in hematological malignancies. Leukemia, 30, 2016

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2016-04-27
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