five

Kynurenine Aminotransferase II Inhibitors

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Protein Data Bank Japan2023-09-13 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4ge4
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资源简介:
Kynurenine Aminotransferase II Inhibitors Descriptor: (5-hydroxy-4-{[(1-hydroxy-7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)amino]methyl}-6-methylpyridin-3-yl)methyl dihydrogen phosphate, Kynurenine/alpha-aminoadipate aminotransferase, mitochondrial Authors: Pandit, J. Deposit date: 2012-08-01 Release date: 2012-11-07 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (2.41 Å) Cite: Structure-Based Design of Irreversible Human KAT II Inhibitors: Discovery of New Potency-Enhancing Interactions. ACS Med Chem Lett, 4, 2013
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2012-08-01
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