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Pim1 in complex with 4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acid and Pimtide

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Protein Data Bank Japan2024-11-13 更新2026-04-19 收录
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Pim1 in complex with 4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acid and Pimtide Descriptor: 4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acid, Pimtide, Serine/threonine-protein kinase pim-1 Authors: Hochban, P.M.M, Heine, A, Diederich, W.E. Deposit date: 2022-07-18 Release date: 2023-02-01 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.15 Å) Cite: Pose, duplicate, then elaborate: Steps towards increased affinity for inhibitors targeting the specificity surface of the Pim-1 kinase. Eur.J.Med.Chem., 245, 2023
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2022-07-18
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