Inhibitor of HIV protease with unusual binding mode potently inhibiting multi-resistant protease mutants
收藏Protein Data Bank Japan2023-10-25 更新2026-03-21 收录
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Inhibitor of HIV protease with unusual binding mode potently inhibiting multi-resistant protease mutants Descriptor: proteinase, {(1S)-1-BENZYL-4-[3-CARBAMOYL-1-(1-CARBAMOYL-2-PHENYL-ETHYLCARBAMOYL)-(S)-PROPYLCARBAMOYL]-2-OXO-5-PHENYL-PENTYL}-CARBAMIC ACID TERT-BUTYL ESTER Authors: Weber, J, Mesters, J.R, Lepsik, M, Prejdova, J, Svec, M, Sponarova, J, Mlcochova, P, Skalicka, K, Strisovsky, K, Uhlikova, T, Soucek, M, Machala, L, Stankova, M, Vondrasek, J, Klimkait, T, Kraeusslich, H.-G, Hilgenfeld, R, Konvalinka, J. Deposit date: 2002-10-02 Release date: 2002-12-23 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Unusual Binding Mode of an HIV-1 Protease Inhibitor Explains its Potency against Multi-drug-resistant Virus Strains J.MOL.BIOL., 324, 2002
创建时间:
2002-10-02



