Tankyrase-1 complexed with small molecule inhibitor
收藏Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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Tankyrase-1 complexed with small molecule inhibitor Descriptor: 4-tert-butyl-N-(5,6-dihydro[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl)benzamide, SULFATE ION, Tankyrase-1, ... Authors: Stams, T, Kirby, C. Deposit date: 2013-05-17 Release date: 2013-08-28 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (2.29 Å) Cite: Structure-Efficiency Relationship of [1,2,4]Triazol-3-ylamines as Novel Nicotinamide Isosteres that Inhibit Tankyrases. J.Med.Chem., 56, 2013
创建时间:
2013-05-17



