Crystal structure of ERK2 complexed with allosteric and ATP-competitive inhibitors.
收藏Protein Data Bank Japan2023-11-08 更新2026-03-21 收录
下载链接：
https://pdbj.org/mine/summary/5ax3
下载链接
链接失效反馈官方服务：
资源简介：
Crystal structure of ERK2 complexed with allosteric and ATP-competitive inhibitors. Descriptor: (2R,3R,4S,5R)-2-(4-AMINO-5-IODO-7H-PYRROLO[2,3-D]PYRIMIDIN-7-YL)-5-(HYDROXYMETHYL)TETRAHYDROFURAN-3,4-DIOL, Mitogen-activated protein kinase 1, allosteric and ATP-competitive inhibitor Authors: Kinoshita, T, Sugiyama, H, Mori, Y, Takahashi, N, Tomonaga, A. Deposit date: 2015-07-14 Release date: 2016-02-10 Last modified: 2023-11-08 Method: X-RAY DIFFRACTION (2.984 Å) Cite: Identification of allosteric ERK2 inhibitors through in silico biased screening and competitive binding assay Bioorg.Med.Chem.Lett., 26, 2016
创建时间：
2015-07-14
