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Human KIF18A-DARPin fusion protein bound to AMP-PNP and tubulin

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Protein Data Bank Japan2025-12-03 更新2026-05-24 收录
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Human KIF18A-DARPin fusion protein bound to AMP-PNP and tubulin Descriptor: 1,2-ETHANEDIOL, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ... Authors: Lockbaum, G.J, Lee, Y.-T, Boriack-Sjodin, P.A, Grigoriu, S. Deposit date: 2025-10-09 Release date: 2025-11-05 Last modified: 2025-12-03 Method: X-RAY DIFFRACTION (2.406 Å) Cite: Discovery of Kinesin KIF18A Inhibitor ATX020: Tactical Application of Silicon Atom Replacement. Acs Med.Chem.Lett., 16, 2025

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2025-10-09
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