1,4-Oxazine BACE1 inhibitors
收藏Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5clm
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资源简介:
1,4-Oxazine BACE1 inhibitors Descriptor: Beta-secretase 1, CHLORIDE ION, IODIDE ION, ... Authors: Rombouts, F, Tresadern, G, Delgado, O, Martinez Lamenca, C, Van Gool, M, Garcia-Molina, A, Alonso De Diego, S, Oehlrich, D, Prokopcova, H, Alonso, J.M, Austin, N, Borghys, H, Van Brandt, S, Surkyn, M, De Cleyn, M, Vos, A, Alexander, R, MacDonald, G, Moechars, D, Trabanco, A, Gijsen, H. Deposit date: 2015-07-16 Release date: 2015-09-30 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.61 Å) Cite: 1,4-Oxazine beta-Secretase 1 (BACE1) Inhibitors: From Hit Generation to Orally Bioavailable Brain Penetrant Leads. J.Med.Chem., 58, 2015
创建时间:
2015-07-16



