Crystal Structure of BRD4(1) bound to inhibitor BUX5 (11)
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Crystal Structure of BRD4(1) bound to inhibitor BUX5 (11) Descriptor: Bromodomain-containing protein 4, ~{N}-(2-methoxy-5-piperidin-1-ylsulfonyl-phenyl)-3-methyl-4-oxidanylidene-5,6,7,8-tetrahydro-2~{H}-cyclohepta[c]pyrrole-1-carboxamide Authors: Huegle, M. Deposit date: 2019-07-16 Release date: 2020-12-09 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.5 Å) Cite: 4-Acyl Pyrroles as Dual BET-BRD7/9 Bromodomain Inhibitors Address BETi Insensitive Human Cancer Cell Lines. J.Med.Chem., 63, 2020
创建时间:
2019-07-16



